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February 2011
Osman, Khadijo and Evangelopoulos, Dimitrios and Basavannacharya, Chandrakala and Gupta, Antima and McHugh, T.D. and Bhakta, Sanjib and Gibbons, S. (2011) An antibacterial from Hypericum acmosepalum inhibits ATP-dependent MurE ligase from Mycobacterium tuberculosis. International Journal of Antimicrobial Agents 39 (2), pp. 124-129. ISSN 0924-8579.
August 2011
Guzman, Juan D. and Wube, A. and Evangelopoulos, Dimitrios and Gupta, Antima and Hufner, A. and Basavannacharya, Chandrakala and Rahman, M.M. and Thomaschitz, C. and Bauer, R. and McHugh, T.D. and Nobeli, Irene and Prieto, J.M. and Gibbons, S. and Bucar, F. and Bhakta, Sanjib (2011) Interaction of N-methyl-2-alkenyl-4-quinolones with ATP-dependent MurE ligase of Mycobacterium tuberculosis: antibacterial activity, molecular docking and inhibition kinetics. Journal of Antimicrobial Chemotherapy 66 (8), pp. 1766-1772. ISSN 0305-7453.
2012
Kottakota, S.K. and Benton, M. and Evangelopoulos, Dimitrios and Guzman, Juan D. and Bhakta, Sanjib and McHugh, T.D. and Gray, M. and Groundwater, P.W. and Marrs, E.C.L. and Perry, J.D. and Harburn, J.J. (2012) Versatile routes to marine sponge metabolites through Benzylidene Rhodanines. Organic Letters 14 (24), pp. 6310-6313. ISSN 1523-7060.
June 2013
Guzman, Juan D. and Evangelopoulos, Dimitrios and Gupta, Antima and Birchall, K. and Mwaigwisya, S. and Saxty, B. and McHugh, T.D. and Gibbons, S. and Malkinson, J. and Bhakta, Sanjib (2013) Antitubercular specific activity of ibuprofen and the other 2-arylpropanoic acids using the HT-SPOTi whole-cell phenotypic assay. BMJ Open 3 (6), e002672. ISSN 2044-6055.
1 May 2014
McGuigan, C. and Derudas, M. and Gonczy, B. and Hinsinger, K. and Kandil, S. and Pertusati, F. and Serpi, M. and Snoeck, R. and Andrei, G. and Balzarini, J. and McHugh, T.D. and Maitra, A. and Akorli, E. and Evangelopoulos, Dimitrios and Bhakta, Sanjib (2014) ProTides of N–(3-(5-(2’-deoxyuridine))prop-2- ynyl)octanamide as potential anti-tubercular and anti-viral agents. Bioorganic & Medicinal Chemistry 22 (9), pp. 2816-2824. ISSN 1464-3391.
April 2015
Hochfellner, C. and Evangelopoulos, Dimitrios and Zloh, M. and Wube, A. and Guzman, J.D. and McHugh, T.D. and Kunert, O. and Bhakta, Sanjib and Bucar, F. (2015) Antagonistic effects of indoloquinazoline alkaloids on antimycobacterial activity of evocarpine. Journal of Applied Microbiology 118 (4), pp. 864-872. ISSN 1364-5072.
11 May 2016
Brucoli, F. and Guzman, Juan David and Basher, M.A. and Evangelopoulos, Dimitrios and Mcmahon, Eleanor and Munshi, Tulika and McHugh, T.D. and Fox, K.R. and Bhakta, Sanjib (2016) DNA sequence-selective C8-linked pyrrolobenzodiazepine–heterocyclic polyamide conjugates show anti-tubercular-specific activities. The Journal of Antibiotics 69 , pp. 843-849. ISSN 0021-8820.
June 2016
Maitra, Arundhati and Bates, S. and Shaik, M. and Evangelopoulos, Dimitrios and Abubakar, I. and McHugh, T.D. and Lipman, M. and Bhakta, Sanjib (2016) Repurposing drugs for treatment of tuberculosis: a role for non-steroidal anti-inflammatory drugs. British Medical Bulletin 118 (1), pp. 138-148. ISSN 1471-8391.
July 2017
Ryan, A. and Polycarpou, E. and Lack, N.A. and Evangelopoulos, Dimitrios and Sieg, C. and Halman, A. and Bhakta, Sanjib and Eleftheriadou, O. and McHugh, T.D. and Keany, S. and Lowe, E.D. and Ballet, R. and Abuhammad, A. and Jacobs, W.R. and Ciulli, A. and Sim, E. (2017) Investigation of the mycobacterial enzyme HsaD as a potential novel target for anti-tubercular agents using a fragment-based drug design approach. British Journal of Pharmacology 174 (14), pp. 2209-2224. ISSN 0007-1188.
18 January 2018
Danquah, C.A. and Kakagianni, E. and Khondkar, P. and Maitra, Arundhati and Rahman, M. and Evangelopoulos, D. and McHugh, T.D. and Stapleton, P. and Malkinson, J. and Bhakta, Sanjib and Gibbons, Simon (2018) Analogues of Disulfides from Allium stipitatum demonstrate potent anti-tubercular activities through drug efflux pump and Biofilm inhibition. Scientific Reports 8 (1), p. 1150. ISSN 2045-2322.
29 March 2018
Schwenk, S. and Moores, A. and Nobeli, Irene and McHugh, T.D. and Arnvig, K.B. (2018) Cell-wall synthesis and ribosome maturation are co-regulated by an RNA switch in Mycobacterium tuberculosis. Nucleic Acids Research , ISSN 0305-1048.
November 2020
Maitra, A. and Evangelopoulos, D. and Chrzastek, A. and Martin, L.T. and Hanrath, A. and Chapman, E. and Hailes, H.C. and Lipman, M. and McHugh, T.D. and Waddell, S.J. and Bhakta, Sanjib (2020) Carprofen elicits pleiotropic mechanisms of bactericidal action with the potential to reverse antimicrobial drug resistance in tuberculosis. The Journal of Antimicrobial Chemotherapy 75 (11), pp. 3194-3201. ISSN 1460-2091.