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Ryan, A. and Polycarpou, E. and Lack, N.A. and Evangelopoulos, Dimitrios and Sieg, C. and Halman, A. and Bhakta, Sanjib and Eleftheriadou, O. and McHugh, T.D. and Keany, S. and Lowe, E.D. and Ballet, R. and Abuhammad, A. and Jacobs, W.R. and Ciulli, A. and Sim, E. (2017) Investigation of the mycobacterial enzyme HsaD as a potential novel target for anti-tubercular agents using a fragment-based drug design approach. British Journal of Pharmacology 174 (14), pp. 2209-2224. ISSN 0007-1188.

Evangelopoulos, Dimitrios and Gupta, Antima and Lack, N. and Maitra, Arundhati and ten Bokum, A.M.C. and Kendall, Sharon L. and Sim, E. and Bhakta, Sanjib (2014) Characterisation of a putative AraC transcriptional regulator from Mycobacterium smegmatis. Tuberculosis 94 (6), pp. 664-671. ISSN 1472-9792.

Evangelopoulos, Dimitrios and Cronin, Nora and Daviter, Tina and Sim, E. and Keep, Nicholas H. and Bhakta, Sanjib (2011) Characterization of an oxidoreductase from the arylamine N-acetyltransferase operon in Mycobacterium Smegmatis. FEBS Journal 278 (24), pp. 4824-4832. ISSN 1742-464X.

Westwood, I.M. and Bhakta, Sanjib and Russell, A.J. and Fullam, E. and Anderton, M.C. and Akane Kawamura, A. and Mulvaney, A.W. and Vickers, R.J. and Bhowruth, V. and Besra, G.S. and Lalvani, A. and Davies, S.G. and Sim, E. (2010) Identification of arylamine N-acetyltransferase inhibitors as an approach towards novel anti-tuberculars. Protein & Cell 1 (1), pp. 82-95. ISSN 1674-800X.

Sim, E. and Sandy, J. and Evangelopoulos, Dimitrios and Fullam, E. and Bhakta, Sanjib and Westwood, I.M. and Krylova, A. and Lack, N. and Noble, M. (2008) Arylamine N-acetyltransferases in mycobacteria. Current Drug Metabolism 9 (6), pp. 510-519. ISSN 1389-2002.

Smellie, I. and Bhakta, Sanjib and Sim, E. and Fairbanks, A. (2007) Synthesis of putative chain terminators of mycobacterial arabinan biosynthesis. Organic and Biomolecular Chemistry 5 (14), pp. 2257-2266. ISSN 1477-0520.

Anderton, M.C. and Bhakta, Sanjib and Besra, G.S. and Jeavons, P. and Eltis, L.D. and Sim, E. (2006) Characterization of the putative operon containing arylamine n-acetyltransferase (nat) in mycobacterium bovis BCG. Molecular Microbiology 59 (1), pp. 181-192. ISSN 0950-382X.

Westwood, I.M. and Holton, S.J. and Rodrigues-Lima, F. and Dupret, J.M. and Bhakta, Sanjib and Noble, M.E. and Sim, E. (2005) Expression, purification, characterization and structure of pseudomonas aeruginosa arylamine N-acetyltransferase. Biochemical Journal 385 (2), pp. 605-612. ISSN 0264-6021.

Bhakta, Sanjib and Besra, G.S. and Upton, A.M. and Parish, T. and Sholto-Douglas-Vernon, C. and Gibson, K.J. and Knutton, S. and Gordon, S. and DaSilva, R.P. and Anderton, M.C. and Sim, E. (2004) Arylamine N-acetyltransferase is required for synthesis of mycolic acids and complex lipids in Mycobacterium bovis BCG and represents a novel drug target. The Journal of Experimental Medicine 199 (9), pp. 1191-1199. ISSN 0022-1007.

Sim, E. and Pinter, K. and Mushtaq, A. and Upton, A. and Sandy, J. and Bhakta, Sanjib and Noble, M. (2003) Arylamine N-acetyltransferases: a pharmacogenomic approach to drug metabolism and endogenous function. Biochemical Society Transactions 31 (3), pp. 615-619. ISSN 0300-5127.

Book Section

Evangelopoulos, Dimitrios and Bhakta, Sanjib (2018) Arylamine N-Acetyltransferase in Mycobacteria. In: Laurieri, N. and Sim, E. (eds.) Arylamine N-acetyltransferases in Health and Disease: From Pharmacogenetics to Drug Discovery and Diagnostics. World Scientific, pp. 303-324. ISBN 9789813232006.